Microorganism |
MIC50 (μg/ml) |
MIC90 (μg/ml) |
Range (μg/ml) |
Antimicrobial  |
Reference |
Staphylococcus aureus (42) |
- |
- |
4 - ? |
CB-182107  |
541 |
Staphylococcus aureus (42) |
- |
- |
4 - ? |
CB-182286  |
541 |
Staphylococcus aureus (42) |
- |
- |
8 - ? |
CB-182130  |
541 |
Staphylococcus aureus (42) |
- |
- |
8 - ? |
CB-182257  |
541 |
Staphylococcus aureus (42) |
- |
- |
16 - ? |
CB-182263  |
541 |
Staphylococcus aureus (42) |
- |
- |
32 - ? |
CB-182251  |
541 |
Staphylococcus aureus (42) |
- |
- |
128 - ? |
CB-182269  |
541 |
Staphylococcus aureus (420 + lincosamide-resistant + macrolide-resistant + streptrogrami) |
- |
- |
? - >50 |
Gentamicin (Gentamycin, Garamycin)  |
68 |
Staphylococcus aureus (420 + macrolide-resistant + lincosamide-resistant + streptrogrami) |
- |
- |
? - 25 |
Tetracycline (Sumycin, Achromycin V, Steclin)  |
68 |
Staphylococcus aureus (425 + linezolid-resistant) |
- |
- |
0.12 - ? |
Oxacillin (Prostaphilin, Bactocil, Prostaphlin)  |
192 |
Staphylococcus aureus (425 + linezolid-resistant) |
- |
- |
1 - ? |
Penicillin (Benzylpenicillin, Penicillin G, Bicillin C-R/L-A, Pfizerpen, Wycellin)  |
192 |
Staphylococcus aureus (425 + linezolid-resistant) |
- |
- |
2 - ? |
Vancomycin (Vancocyn, Lyphocin)  |
192 |
Staphylococcus aureus (425 + linezolid-resistant) |
- |
- |
8 - ? |
TR-700  |
192 |
Staphylococcus aureus (425 + linezolid-resistant) |
- |
- |
32 - ? |
Linezolid (PNU-100766, U-100766, Zyvox)  |
192 |
Staphylococcus aureus (4280-0256 + methicillin-resistant) |
- |
- |
4 - ? |
RWJ-416457  |
280 |
Staphylococcus aureus (4319 + methicillin-susceptible + ESBL) |
- |
- |
0.094 - ? |
Penicillin (Benzylpenicillin, Penicillin G, Bicillin C-R/L-A, Pfizerpen, Wycellin)  |
1055 |
Staphylococcus aureus (4319 + methicillin-susceptible + ESBL) |
- |
- |
0.75 - ? |
Oxacillin (Prostaphilin, Bactocil, Prostaphlin)  |
1055 |
Staphylococcus aureus (450 + methicillin-resistant) |
- |
- |
>16 - ? |
Ciprofloxacin (Cipro, Ciproxin, Ciprobay)  |
180 |
Staphylococcus aureus (4698 + methicillin-resistant) |
- |
- |
? - >50 |
Gentamicin (Gentamycin, Garamycin)  |
68 |
Staphylococcus aureus (4698 + methicillin-resistant) |
- |
- |
? - >50 |
Tetracycline (Sumycin, Achromycin V, Steclin)  |
68 |
Staphylococcus aureus (4699 + methicillin-resistant) |
- |
- |
? - >50 |
Gentamicin (Gentamycin, Garamycin)  |
68 |
Staphylococcus aureus (4699 + methicillin-resistant) |
- |
- |
? - >50 |
Tetracycline (Sumycin, Achromycin V, Steclin)  |
68 |
Staphylococcus aureus (480 + linezolid-resistant) |
- |
- |
<0.03 - ? |
Oxacillin (Prostaphilin, Bactocil, Prostaphlin)  |
192 |
Staphylococcus aureus (480 + linezolid-resistant) |
- |
- |
0.25 - ? |
Penicillin (Benzylpenicillin, Penicillin G, Bicillin C-R/L-A, Pfizerpen, Wycellin)  |
192 |
Staphylococcus aureus (480 + linezolid-resistant) |
- |
- |
1 - ? |
Vancomycin (Vancocyn, Lyphocin)  |
192 |
Staphylococcus aureus (480 + linezolid-resistant) |
- |
- |
16 - ? |
TR-700  |
192 |
Staphylococcus aureus (480 + linezolid-resistant) |
- |
- |
>32 - ? |
Linezolid (PNU-100766, U-100766, Zyvox)  |
192 |
Staphylococcus aureus (494 + methicillin-resistant) |
- |
- |
0.008 - ? |
Rifampicin (Rifampin)  |
235 |